Rational design and validation of a Tip60 histone acetyltransferase inhibitor

Chunxia Gao, Emer Bourke, Martin Scobie, Melina Arcos Famme, Tobias Koolmeister, Thomas Helleday, Leif A. Eriksson, Noel F. Lowndes, James A.L. Brown

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Biochemistry, Genetics and Molecular Biology